SCHEMBL6206465

SCHEMBL6206465

O=C1N=COC1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.40
CTRB1 P17538 1/20 0.38
CES2 O00748 2/20 0.37
FASN P49327 1/20 0.37
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
EP300 Q09472 1/20 0.35
MAOB P27338 1/20 0.35
GRM2 Q14416 1/20 0.35
MDM2 Q00987 4/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5967437 1.00 TLR9 (0.40) TLR9CTRB1CES2FASNLMNA
SCHEMBL11741164 0.86 LTA4H (0.41) LMNA
SCHEMBL11737987 0.84 NOTUM (0.39) LMNAGAA
SCHEMBL11454739 0.82 FASN (0.41) FASN
SCHEMBL11739217 0.82 GAA (0.40) CES2LMNAGAAMDM2
SCHEMBL11740374 0.82 MDM2 (0.38) LMNAGAAMAOBGRM2MDM2
SCHEMBL11741970 0.82 MDM2 (0.40) CES2LMNAGAAMDM2
SCHEMBL11741375 0.80 TAAR1 (0.38) MAOB
SCHEMBL11743542 0.80 LPL (0.37) LMNAGAA
SCHEMBL11737101 0.78 DPP4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-52007959-A None JP disclosed
JP-52031071-A None JP disclosed
JP-52048663-A None JP disclosed
EP-1503997-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2005-02-09 EP disclosed
WO-2003097617-A1 CYSTEINE PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2003-11-27 WO disclosed
CN-1143960-A Therapeutic heterocyclic compounds WELLCOME FOUND (GB) 1997-02-26 CN disclosed
US-5545568-A ARRAY OF COMPOUNDS ON SUBSTRATE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-08-13 US disclosed
WO-1994006291-A1 SOLID PHASE AND COMBINATORIAL SYNTHESIS OF COMPOUNDS ON A SOLID SUPPORT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-03-31 WO disclosed
US-5288514-A Linking a protected 2-aminobenzophenone to a substrate; deprotecting and reacting with an amino acid; cyclization; removal from substrate; screening THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-02-22 US disclosed
US-4062862-A MUSCLE RELAXANT NIPPON CHEMIPHAR CO., LTD. (JA) 1977-12-13 US disclosed
US-4062862-A MUSCLE RELAXANT NIPPON CHEMIPHAR CO., LTD. (JA) 1977-12-13 US disclosed
US-4062862-A MUSCLE RELAXANT NIPPON CHEMIPHAR CO., LTD. (JA) 1977-12-13 US disclosed
JP-S5248663-A PREPARATION OF 5-BENZYL-2-OXAZOLIDONE DERIVATIVES NIPPON CHEMIPHAR CO LTD 1977-04-18 JP disclosed
JP-S5231071-A 5-BENZYL-2-OXAZOLIDONE DERIVATIVES NIPPON CHEMIPHAR CO LTD 1977-03-09 JP disclosed
JP-S527959-A PREPARATION OF 5-BENZYL-2-OXAZOLIDONE DERIVATIVES NIPPON CHEMIPHAR CO LTD 1977-01-21 JP disclosed