SCHEMBL6206773

SCHEMBL6206773

CCCCCCCCNC(=O)Nc1sc(C(=O)NCCc2cccnc2)c(CC)c1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.42
FAAH O00519 1/20 0.40
FLT4 P35916 2/20 0.39
FES P07332 1/20 0.39
RET P07949 1/20 0.39
MARK3 P27448 1/20 0.39
TYK2 P29597 1/20 0.39
SYK P43405 1/20 0.39
CLK2 P49760 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
PTAFR P25105 5/20 0.38
CHRM4 P08173 1/20 0.38
CDK2 P24941 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TRPV1 Q8NER1 1/20 0.37
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6030971 0.91 ALDH1A1 (0.44) CYP3A4FAAHFLT4FESRET
SCHEMBL6029645 0.84 ALDH1A1 (0.49) CYP3A4FAAHFLT4FESRET
SCHEMBL6030084 0.81 CHRM4 (0.45) FAAHFLT4FESRETMARK3
SCHEMBL16643981 0.78 ALDH1A1 (0.59) CYP3A4ALDH1A1KDM4EMEN1LMNA
SCHEMBL6030667 0.78 NPC1 (0.46) CYP3A4ALDH1A1KDM4EMEN1LMNA
SCHEMBL6030651 0.78 NPC1 (0.46) CYP3A4ALDH1A1KDM4EMEN1GAA
SCHEMBL6031608 0.77 ALDH1A1 (0.47) CYP3A4FAAHFLT4CDK2ALDH1A1
SCHEMBL6029757 0.76 ALDH1A1 (0.43) ALDH1A1KDM4EMEN1LMNAMAPT
SCHEMBL6030054 0.76 ALDH1A1 (0.43) ALDH1A1KDM4EMEN1LMNAMAPT
SCHEMBL6029710 0.76 ALDH1A1 (0.43) ALDH1A1KDM4EMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1467978-A4 PANCREATIC LIPASE INHIBITOR COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2005-11-02 EP disclosed
EP-1467978-A1 PANCREATIC LIPASE INHIBITOR COMPOUNDS, THEIR SYNTHESIS AND USE OSI Pharmaceuticals, Inc. (US) 2004-10-20 EP disclosed
WO-2003053944-A1 PANCREATIC LIPASE INHIBITOR COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARMACEUTICALS, INC. (US) 2003-07-03 WO disclosed