SCHEMBL6206862

SCHEMBL6206862

N#Cc1ccc2nccc(CCN3CC[CH][C@@H](O)C3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.38
CDK8 P49336 8/20 0.38
CCNC P24863 5/20 0.38
KCNH2 Q12809 4/20 0.36
KCNJ1 P48048 1/20 0.36
CDK19 Q9BWU1 3/20 0.36
MAP4K2 Q12851 1/20 0.36
HASPIN Q8TF76 1/20 0.36
IRAK4 Q9NWZ3 3/20 0.36
DRD2 P14416 3/20 0.36
DRD3 P35462 3/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4480929 0.81 HRH3 (0.38) CDK8CCNCKCNH2CDK19MAP4K2
SCHEMBL5305790 0.77 CCR5 (0.43) SLC22A12CDK8CCNCKCNH2CDK19
SCHEMBL4497675 0.77 DRD2 (0.39) SLC22A12CDK8CCNCKCNH2CDK19
SCHEMBL4497667 0.77 DRD2 (0.39) SLC22A12CDK8CCNCKCNH2CDK19
SCHEMBL5308578 0.76 KCNH2 (0.49) CDK8CCNCKCNH2KCNJ1IRAK4
SCHEMBL5305787 0.73 CCR3 (0.42) SLC22A12CDK8CCNCKCNH2CDK19
SCHEMBL3400497 0.73 CDK8 (0.49) SLC22A12CDK8CCNCCDK19IRAK4
SCHEMBL14610965 0.71 CDK8 (0.42) CDK8CCNCKCNH2CDK19MAP4K2
SCHEMBL4495204 0.70 DRD2 (0.51) CDK8CCNCKCNH2IRAK4DRD2
SCHEMBL13921377 0.69 KCNH2 (0.48) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583537-A3 PIPERIDINE COMPOUNDS AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2005-12-14 EP disclosed
EP-1583537-A2 PIPERIDINE COMPOUNDS AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2005-10-12 EP disclosed
WO-2004002490-A2 PIPERIDINE COMPOUNDS AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2004-01-08 WO disclosed