SCHEMBL6207925

SCHEMBL6207925

NC(=O)CCC(=O)c1nc(C2CC2)no1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
LDHA P00338 2/20 0.32
HSD11B1 P28845 1/20 0.32
CA12 O43570 1/20 0.32
POLB P06746 1/20 0.32
CASP3 P42574 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
AKR1C4 P17516 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
SMYD3 Q9H7B4 1/20 0.31
FABP4 P15090 2/20 0.31
FABP5 Q01469 2/20 0.31
AOC3 Q16853 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433614 0.80 CA1 (0.40) CA1CA2CA9LDHAHSD11B1
SCHEMBL5955867 0.76 CA1 (0.33) CA1CA2CA9LDHAHSD11B1
SCHEMBL17898050 0.73 PIK3CG (0.36) CA1CA2CA9LDHAHSD11B1
SCHEMBL27365749 0.71 AKR1C4 (0.42) HSD11B1POLBCASP3SENP7SENP6
SCHEMBL5955871 0.70 DPP4 (0.37) CA1CA2CA9DPP4DPP8
SCHEMBL17897216 0.69 FABP4 (0.36) CA1CA2CA9HSD11B1POLB
SCHEMBL5516375 0.68 SMN1; SMN2 (0.32) CA1CA2CA9HSD11B1POLB
SCHEMBL5516368 0.68 SMN1; SMN2 (0.32) CA1CA2CA9HSD11B1POLB
SCHEMBL14427060 0.65 FABP4 (0.33) LDHAHSD11B1POLBFABP4FABP5
SCHEMBL14110444 0.64 CPT1A (0.37) LDHAHSD11B1POLBAKR1C4AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515726-A1 MORPHOLINE AND TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS CATHEPSIN INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2005-03-23 EP claimed
WO-2004002491-A1 MORPHOLINE AND TETRAHYDROPYRAN DRIVATIVES AND THEIR USE AS CATHEPSIN INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2004-01-08 WO claimed