SCHEMBL6208729

SCHEMBL6208729

CC(C)CC(NC(=O)c1ccc(N2CCNCC2)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cc[nH]c(=O)c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.49
CTSS P25774 1/20 0.39
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
ITGA2 P17301 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041438 0.90 CTSK (0.56) CTSKCTSSADRB2ADRB1ADRB3
SCHEMBL6214663 0.89 CTSK (0.51) CTSKCTSSSMYD3
SCHEMBL4042258 0.88 CTSK (0.51) CTSKCTSSADRB2ADRB1ADRB3
SCHEMBL4046529 0.87 CTSK (0.49) CTSKCTSSADRB2ADRB1ADRB3
SCHEMBL6209624 0.87 CTSK (0.59) CTSKCTSSITGB3ITGA2BITGA2
SCHEMBL4045775 0.86 CTSK (0.49) CTSKCTSSADRB2ADRB1ADRB3
SCHEMBL4044861 0.86 CTSK (0.49) CTSKCTSSADRB2ADRB1ADRB3
SCHEMBL6210948 0.84 CTSK (0.48) CTSKCTSS
SCHEMBL4041465 0.83 CTSK (0.51) CTSKCTSS
SCHEMBL4045440 0.83 CTSK (0.59) CTSKCTSSADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed