SCHEMBL6209624

SCHEMBL6209624

CC(C)CC(NC(=O)c1ccc(N2CCNCC2)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1cc[nH]c(=O)c1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.59
CTSS P25774 3/20 0.46
SMYD3 Q9H7B4 1/20 0.40
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ITGA2 P17301 1/20 0.36
CDK4 P11802 1/20 0.35
CCNA2 P20248 1/20 0.35
CCND1 P24385 1/20 0.35
CDK2 P24941 1/20 0.35
CTSL P07711 2/20 0.35
CTSB P07858 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6211024 0.93 CTSK (0.60) CTSKCTSS
SCHEMBL4044020 0.88 CTSK (0.75) CTSKCTSSITGB3ITGA2BCDK4
SCHEMBL5941816 0.88 CTSK (0.75) CTSKCTSSITGB3ITGA2BCDK4
SCHEMBL4368915 0.88 CTSK (0.75) CTSKCTSSITGB3ITGA2BCDK4
SCHEMBL6209777 0.88 CTSK (0.63) CTSKCTSSSMYD3
SCHEMBL4368912 0.88 CTSK (0.75) CTSKCTSSITGB3ITGA2BCDK4
SCHEMBL4040434 0.87 CTSK (0.64) CTSKCTSSCDK4CCNA2CCND1
SCHEMBL6208729 0.87 CTSK (0.49) CTSKCTSSSMYD3ITGB3ITGA2B
SCHEMBL4038951 0.86 CTSK (0.57) CTSKCTSSITGB3ITGA2BCDK4
SCHEMBL4038247 0.86 CTSK (0.59) CTSKCTSSSMYD3ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed