SCHEMBL6209065

SCHEMBL6209065

CN1CCN(c2ccc(C(=O)NCCCCC(=O)N3CCC4C3C(=O)CN4S(=O)(=O)Cc3ccccn3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.43
HDAC3 O15379 3/20 0.43
DRD3 P35462 5/20 0.38
HTR1A P08908 3/20 0.38
HTR2A P28223 3/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
ADRA1B P35368 1/20 0.38
KCNH2 Q12809 1/20 0.38
DRD2 P14416 4/20 0.38
DRD4 P21917 2/20 0.38
NAMPT P43490 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.36
KDM1A O60341 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6209329 0.92 HDAC3 (0.42) HDAC1HDAC3DRD3HTR1AHTR2A
SCHEMBL6262865 0.89 HDAC3 (0.45) HDAC1HDAC3DRD3HTR1AHTR2A
SCHEMBL6210338 0.87 DPP4 (0.46) HDAC1HDAC3DRD3DRD4NAMPT
SCHEMBL6210861 0.87 HDAC1 (0.41) HDAC1HDAC3DRD3HTR1AHTR2A
SCHEMBL6211778 0.83 TAOK1 (0.37) DRD3DRD2NAMPTNPC1GAA
SCHEMBL6212649 0.83 NPC1 (0.40) DRD3DRD2NAMPTNPC1GAA
SCHEMBL4039077 0.82 CTSK (0.57)
SCHEMBL4040968 0.81 CTSK (0.47)
SCHEMBL6211482 0.80 HDAC3 (0.40) HDAC1HDAC3DRD3DRD2HDAC8
SCHEMBL6210120 0.80 GAA (0.38) NAMPTNPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed