SCHEMBL6211482

SCHEMBL6211482

CN1CCN(c2ccc(C(=O)NCCCCC(=O)N3CCC4C3C(=O)CN4S(=O)(=O)C3=NC=CCC3=O)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 11/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC8 Q9BY41 9/20 0.36
VDR P11473 2/20 0.36
CTSK P43235 1/20 0.35
DPP4 P27487 1/20 0.35
DRD3 P35462 2/20 0.34
MAPK14 Q16539 1/20 0.34
DRD2 P14416 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6210811 0.85 CHRM4 (0.40) DPP4DRD3DRD2
SCHEMBL6210064 0.84 CHRM2 (0.39) HDAC3HDAC1DPP4DRD3DRD2
SCHEMBL6262865 0.83 HDAC3 (0.45) HDAC3HDAC1HDAC8VDRDRD3
SCHEMBL6210241 0.83 ROCK2 (0.36) HDAC3HDAC1HDAC8DPP4HDAC6
SCHEMBL6213828 0.82 CTSK (0.57) CTSK
SCHEMBL6209065 0.80 HDAC1 (0.43) HDAC3HDAC1HDAC8DRD3DRD2
SCHEMBL6210861 0.79 HDAC1 (0.41) HDAC3HDAC1HDAC8DRD3HDAC6
SCHEMBL6209349 0.77
SCHEMBL6259546 0.74 ALDH1A1 (0.46) HDAC3HDAC1DRD3DRD2
SCHEMBL6213962 0.74 CTSK (0.41) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed