SCHEMBL6211129

SCHEMBL6211129

CCC(=O)C(C)CN(C)C.CCC(=O)C(C)CN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.47
KCNH2 Q12809 2/20 0.42
OPRM1 P35372 2/20 0.42
OPRD1 P41143 2/20 0.42
MRGPRX2 Q96LB1 1/20 0.42
CHRM3 P20309 1/20 0.42
HRH2 P25021 1/20 0.42
HTR2A P28223 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRK1 P41145 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
LMNA P02545 1/20 0.41
RORC P51449 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6336428 0.94 HPGD (0.47) HPGDMEN1KMT2AALDH1A1NPC1
SCHEMBL6211134 0.79 HPGD (0.39) HPGDMEN1KMT2AALDH1A1NPC1
SCHEMBL669860 0.77 KCNH2 (0.30) KCNH2OPRM1OPRD1MRGPRX2CHRM3
SCHEMBL15370923 0.77 KCNH2 (0.30) KCNH2OPRM1OPRD1MRGPRX2CHRM3
SCHEMBL668761 0.77 KCNH2 (0.30) KCNH2OPRM1OPRD1MRGPRX2CHRM3
SCHEMBL11240083 0.75 HPGD (0.47) HPGDKCNH2HTR2AMEN1KMT2A
Hydrochloric Acid SCHEMBL6906945 0.75 HTT (0.32) OPRM1OPRD1TSHRNPC1RAB9A
SCHEMBL15688853 0.74 HPGD (0.46) HPGDMEN1KMT2ANPC1RAB9A
SCHEMBL10140576 0.73 KMT2A (0.57) HPGDKCNH2HTR2AADRA1AOPRK1
SCHEMBL19047046 0.73 ALDH1A1 (0.50) HPGDMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507521-A1 METABOLITE OF 1-DIMETHYLAMINO-3-(3-METHOXY-PHENYL)-2-METHYL-PENTANE-3-OL AND THE USE THEREOF IN THE TREATMENT OF URINARY INCONTINENCE Grünenthal GmbH (DE) 2005-02-23 EP disclosed
WO-2003101440-A1 METABOLITE OF 1-DIMETHYLAMINO-3-(3-METHOXY-PHENYL)-2-METHYL-PENTANE-3-OL AND THE USE THEREOF IN THE TREATMENT OF URINARY INCONTINENCE Grünenthal GmbH (DE) 2003-12-11 WO disclosed