SCHEMBL6211368

SCHEMBL6211368

CC(C)C[C@@H](Sc1ccc(-c2ccc(CNCc3ccccc3)cc2)cc1)C(=O)NCC#N

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.55
CTSS P25774 9/20 0.55
CTSB P07858 7/20 0.52
CTSL P07711 8/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4700384 1.00 CTSK (0.55) CTSKCTSSCTSBCTSL
SCHEMBL6211886 0.89 CTSK (0.67) CTSKCTSSCTSBCTSL
SCHEMBL4701868 0.89 CTSK (0.67) CTSKCTSSCTSBCTSL
SCHEMBL4698421 0.88 CTSK (0.51) CTSKCTSSCTSBCTSL
SCHEMBL4699909 0.85 CTSK (0.53) CTSKCTSSCTSBCTSL
SCHEMBL4699985 0.84 CTSK (0.52) CTSKCTSSCTSBCTSL
SCHEMBL6271092 0.84 CTSK (0.52) CTSKCTSSCTSBCTSL
SCHEMBL4701062 0.83 CTSK (0.47) CTSKCTSSCTSBCTSL
SCHEMBL4698876 0.82 CTSS (0.58) CTSKCTSSCTSBCTSL
SCHEMBL4702083 0.81 HRH3 (0.47) CTSKCTSSCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-A4 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2005-10-12 EP disclosed
EP-1372655-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Frosst Canada & Co. (CA) 2004-01-02 EP disclosed
WO-2002069901-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2002-09-12 WO disclosed