SCHEMBL6212802

SCHEMBL6212802

Cc1cc[n+]([O-])c(C)c1C(=O)N1CCC(C)(N2CCC(Nc3ncccc3-c3ccccc3)CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.61
CYP3A4 P08684 1/20 0.59
KCNH2 Q12809 4/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4385620 0.76 CCR5 (1.00) CCR5CYP3A4KCNH2
SCHEMBL619811 0.74 CCR5 (1.00) CCR5CYP3A4KCNH2
SCHEMBL4391363 0.73 CCR5 (0.62) CCR5CYP3A4KCNH2
SCHEMBL3843997 0.71 CCR5 (1.00) CCR5KCNH2
SCHEMBL3837942 0.71 CCR5 (1.00) CCR5CYP3A4KCNH2
SCHEMBL3837456 0.69 CCR5 (0.88) CCR5CYP3A4KCNH2
SCHEMBL3840733 0.68 CCR5 (1.00) CCR5CYP3A4KCNH2
Hydrochloric Acid SCHEMBL4199725 0.67 CCR5 (0.71) CCR5CYP3A4KCNH2
SCHEMBL14024851 0.67 CCR5 (0.84) CCR5CYP3A4KCNH2
SCHEMBL4208021 0.67 CCR5 (0.67) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551827-A1 PIPERIDINE DERIVATIVES AS CCR5 INHIBITORS Novartis AG (CH) 2005-07-13 EP disclosed
WO-2004031172-A1 PIPERIDINE DERIVATIVES AS CCR5 INHIBITORS NOVARTIS AG (CH) 2004-04-15 WO disclosed