SCHEMBL6212907

SCHEMBL6212907

COc1ccc(-n2nc(Cl)cc2-c2cc[c]cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.53
PTGS1 P23219 7/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
CYP2C19 P33261 1/20 0.53
THPO P40225 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
HIF1A Q16665 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MALT1 Q9UDY8 1/20 0.49
RPA1 P27694 2/20 0.49
MARS1 P56192 1/20 0.46
ALOX5 P09917 1/20 0.45
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
CCKAR P32238 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5148696 0.83 PTGS2 (0.56) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5148713 0.83 PTGS2 (0.53) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5148723 0.81 PTGS2 (0.54) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5150623 0.80 PTGS2 (0.53) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5152059 0.79 PTGS2 (0.52) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL7872946 0.79 PTGS2 (0.62) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL6540577 0.78 PTGS2 (0.51) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL5148744 0.77 PTGS2 (0.50) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5147862 0.76 MDM2 (0.59) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5150244 0.76 PTGS2 (0.58) PTGS2PTGS1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567503-A1 PYRAZOLE DERIVATIVES USEFUL AS COX-I INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-08-31 EP disclosed
WO-2004050632-A1 PYRAZOLE DERIVATIVES USEFUL AS COX-I INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-17 WO disclosed