SCHEMBL6217754

SCHEMBL6217754

O=C(O)c1cc2[nH]cncc-2c(=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLK2 Q86UE8 1/20 0.39
CYP3A4 P08684 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
GABRA1 P14867 1/20 0.36
NFKB1 P19838 1/20 0.36
GABRR1 P24046 1/20 0.36
GABRR2 P28476 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.36
IDO1 P14902 9/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.35
PMP22 Q01453 1/20 0.35
ECE1 P42892 1/20 0.35
NAPRT Q6XQN6 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
BLM P54132 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6813952 0.79 CYP3A4 (0.42) CYP3A4ALDH1A1TSHRGABRA1NFKB1
SCHEMBL2564383 0.72 IDO1 (0.47) CYP3A4IDO1
SCHEMBL9275774 0.70 ASIC3 (0.33) CYP3A4IDO1MAPT
SCHEMBL6638123 0.67 CYP3A4 (0.60) CYP3A4ALDH1A1TSHRIDO1KDM4E
SCHEMBL940610 0.67 IDO1 (0.59) CYP3A4IDO1
SCHEMBL12263263 0.67 MKNK1 (0.47) TLK2ALDH1A1TSHRKDM4E
SCHEMBL3008680 0.66 RXRA (0.46) CYP3A4ALDH1A1IDO1KDM4EMAPT
SCHEMBL3141716 0.66 IDO1 (0.44) CYP3A4IDO1
4-Imidazolecarboxylic Acid SCHEMBL317725 0.65
Hydrochloric Acid SCHEMBL11257477 0.65 IDO1 (0.43) CYP3A4IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1361873-A4 MATRIX METALLOPROTEINASE INHIBITORS WARNER LAMBERT CO (US) 2005-10-26 EP disclosed
EP-1361873-A2 MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064080-A2 MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LCC (US) 2002-08-22 WO disclosed