SCHEMBL6218705

SCHEMBL6218705

CC(Nc1nccc(-c2sc(C3CCNCC3)nc2-c2ccc(F)cc2)n1)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.65
ACHE P22303 1/20 0.64
EGFR P00533 1/20 0.60
RAF1 P04049 1/20 0.60
ERBB2 P04626 1/20 0.60
SRC P12931 1/20 0.60
KDR P35968 1/20 0.60
MAPK8 P45983 1/20 0.60
MAPK9 P45984 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6218709 1.00 KCNH2 (0.65) KCNH2ACHEEGFRRAF1ERBB2
SCHEMBL5818632 1.00 KCNH2 (0.65) KCNH2ACHEEGFRRAF1ERBB2
SCHEMBL5813602 0.91 MAPK13 (0.57) KCNH2ACHERAF1MAPK9
SCHEMBL5819638 0.90 KCNH2 (0.53) KCNH2ACHEEGFRRAF1ERBB2
SCHEMBL6488022 0.89 EGFR (0.76) KCNH2EGFRRAF1ERBB2SRC
SCHEMBL6488017 0.89 EGFR (0.76) KCNH2EGFRRAF1ERBB2SRC
SCHEMBL5824185 0.88 MAPK13 (0.51) KCNH2ACHERAF1MAPK9
SCHEMBL5818421 0.86 MAPK13 (0.56) KCNH2ACHERAF1MAPK9
SCHEMBL5820631 0.86 MAPK13 (0.55) KCNH2ACHERAF1MAPK9
SCHEMBL5818883 0.85 KCNH2 (0.79) KCNH2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224185-B1 THIAZOLE AND IMIDAZO[4,5-B]PYRIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USE NOVARTIS AG (CH) 2005-11-30 EP disclosed
US-6608072-B1 Inhibiting production of soluble tumor necrosis factor or reducing inflammation NOVARTIS AG (CH) 2003-08-19 US disclosed