SCHEMBL6222995

SCHEMBL6222995

CC(=O)Oc1cnc2c(-c3cccc(F)c3)nn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c2c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TBXA2R P21731 1/20 0.37
PTGDR Q13258 1/20 0.37
GRIN2B Q13224 4/20 0.37
MAPK1 P28482 1/20 0.36
SLC16A3 O15427 1/20 0.35
SLC16A1 P53985 1/20 0.35
MCTS1 Q9ULC4 1/20 0.35
CSNK1E P49674 1/20 0.35
PTGER1 P34995 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13927631 0.83 ALDH1A1 (0.45) PTGDR2KDM4EALDH1A1TBXA2RPTGDR
SCHEMBL6222657 0.82 PTGER1 (0.39) PTGDR2CSNK1EPTGER1HCRTR1HCRTR2
SCHEMBL4140254 0.76 PDE4A (0.39) KDM4EALDH1A1GRIN2BMAPK1PTGER1
SCHEMBL4146332 0.71 KDM4E (0.45) PTGDR2KDM4ETBXA2RPTGDRCSNK1E
SCHEMBL6223386 0.71 TRPA1 (0.49) PTGDR2KDM4EGRIN2BMAPK1
SCHEMBL2857932 0.71 PTGER1 (0.41) ALDH1A1CSNK1EPTGER1
SCHEMBL27536115 0.70 ALDH1A1 (0.41) KDM4EALDH1A1MAPK1PTGER1
SCHEMBL4145901 0.70 MAPK1 (0.38) KDM4EALDH1A1MAPK1PTGER1
SCHEMBL4137268 0.70 DPP4 (0.42) KDM4EALDH1A1MAPK1CSNK1EPTGER1
SCHEMBL2865256 0.69 PTGER1 (0.41) KDM4EALDH1A1CSNK1EPTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1656079-A Pyrazole compounds and pharmaceutical compositions containing the same EISAI CO LTD (JP) 2005-08-17 CN disclosed
EP-1510516-A1 PYRAZOLE COMPOUND AND MEDICINAL COMPOSITION CONTAINING THE SAME Eisai Co., Ltd. (JP) 2005-03-02 EP disclosed