SCHEMBL6228447

SCHEMBL6228447

COc1ccc(C2C=NNC(=O)C2)cc1OCC1(c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 15/20 0.42
PDE4B Q07343 9/20 0.42
PDE4C Q08493 9/20 0.42
PDE4D Q08499 9/20 0.42
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
ESR2 Q92731 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PDE1C Q14123 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226932 0.85 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6232762 0.83 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DHSD17B10
SCHEMBL6232071 0.82 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPOLB
SCHEMBL6229490 0.81 PDE4A (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL498074 0.81 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6228923 0.78 PDE4A (0.47) PDE4APDE4BPDE4CPDE4D
SCHEMBL6229565 0.78 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6232341 0.78 PDE4A (0.60) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6228237 0.78 PDE4B (0.48) PDE4APDE4BPDE4CPDE4D
SCHEMBL6229342 0.78 PDE4A (0.60) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0933366-B1 5-PHENYL-3-PYRIDAZINONE DERIVATIVES AND DRUG COMPOSITIONS CONTAINING THE SAME NIKKEN CHEMICALS CO LTD (JP) 2005-04-06 EP disclosed
US-6235739-B1 ANTIINFLAMMATORY AGENTS; ANTIHISTAMINES; SKIN DISORDERS NIKKEN CHEMICALS CO., LTD. (JP) 2001-05-22 US disclosed
EP-0933366-A1 5-PHENYL-3-PYRIDAZINONE DERIVATIVES AND DRUG COMPOSITIONS CONTAINING THE SAME Nikken Chemicals Company, Limited (JP) 1999-08-04 EP disclosed