SCHEMBL6229736

SCHEMBL6229736

Nc1cc(-c2ccc(Cl)cc2)ccc1OC(=O)NCCc1ccc(CN2CCC(Oc3ccccn3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
MCHR1 Q99705 6/20 0.41
CHRM1 P11229 2/20 0.41
HTR2A P28223 2/20 0.41
CYP2D6 P10635 1/20 0.41
UTS2R Q9UKP6 2/20 0.40
CXCR3 P49682 1/20 0.40
GPBAR1 Q8TDU6 3/20 0.40
RAB9A P51151 2/20 0.40
AKT1 P31749 1/20 0.40
FFAR1 O14842 1/20 0.40
CHRM4 P08173 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6224533 0.88 FAAH (0.45) NPC1MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6704716 0.88 MCHR1 (0.52) NPC1MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6222465 0.87 AKT1 (0.43) MCHR1CHRM1HTR2ACYP2D6UTS2R
SCHEMBL6226147 0.83 MEN1 (0.51) MCHR1CHRM1HTR2ACYP2D6CXCR3
SCHEMBL6225694 0.82 MCHR1 (0.61) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6226841 0.81 MCHR1 (0.61) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6225461 0.80 MCHR1 (0.47) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6708084 0.79 NPC1 (0.50) NPC1MCHR1CHRM1HTR2ACYP2D6
SCHEMBL6228525 0.79 CCR3 (0.49) MCHR1CHRM1HTR2ACYP2D6CHRM4
SCHEMBL6223456 0.77 MCHR1 (0.52) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534689-A1 NOVEL CARBOXAMIDE COMPOUNDS HAVING AN MCH-ANTAGONISTIC EFFECT, MEDICAMENTS CONTAINING SAID COMPOUNDS, AND METHODS FOR THE PRODUCTION THEREOF BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-06-01 EP disclosed
WO-2004024702-A1 NOVEL CARBOXAMIDE COMPOUNDS HAVING AN MCH-ANTAGONISTIC EFFECT, MEDICAMENTS CONTAINING SAID COMPOUNDS, AND METHODS FOR THE PRODUCTION THEREOF BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-03-25 WO disclosed