SCHEMBL6231022

SCHEMBL6231022

O=C(O)NC(C(=O)N1CCOCC1)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 6/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KCNA5 P22460 1/20 0.44
P2RX7 Q99572 1/20 0.44
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13920469 0.89 ALDH1A1 (0.47) TACR1CYP2C9CYP3A4CYP2C19ALDH1A1
SCHEMBL8337162 0.83 ALDH1A1 (0.49) TACR1CYP2C9CYP3A4CYP2C19ALDH1A1
SCHEMBL4705370 0.79 ALDH1A1 (0.48) CYP2C9CYP3A4CYP2C19ALDH1A1MEN1
SCHEMBL13920467 0.77 FAAH (0.44) NAMPT
SCHEMBL20491159 0.76 TACR1 (0.51) TACR1ALDH1A1MEN1KMT2AKDM4E
SCHEMBL10179506 0.76 ALDH1A1 (0.46) CYP2C9CYP3A4CYP2C19ALDH1A1MEN1
SCHEMBL13374225 0.76 ALDH1A1 (0.46) CYP2C9CYP3A4CYP2C19ALDH1A1MEN1
SCHEMBL11958663 0.76 ALDH1A1 (0.48) CYP2C9CYP3A4CYP2C19ALDH1A1MEN1
SCHEMBL4706451 0.75 ALDH1A1 (0.43) TACR1CYP2C9CYP3A4CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL4210812 0.75 ALDH1A1 (0.47) CYP2C9CYP3A4CYP2C19ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567489-A1 PYRROLIDIN-2-ONE DERIVATIVES AS INHIBITORS OF THROMBIN AND FACTOR XA GLAXO GROUP LIMITED (GB) 2005-08-31 EP disclosed
WO-2004052851-A1 PYRROLYDIN-2-ONE DERIVATIVES AS INHIBITORS OF THROMBIN AND FACTOR XA GLAXO GROUP LIMITED (GB) 2004-06-24 WO disclosed