SCHEMBL6231072

SCHEMBL6231072

COc1ccc(-c2nc(C)oc2-c2ccc(O)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.53
NOX1 Q9Y5S8 1/20 0.50
ESR1 P03372 1/20 0.49
MAPK13 O15264 1/20 0.48
MAPK12 P53778 1/20 0.48
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
MAPT P10636 4/20 0.46
TP53 P04637 2/20 0.46
PTGS2 P35354 5/20 0.46
PPARD Q03181 3/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
APP P05067 1/20 0.45
PTGS1 P23219 2/20 0.45
LTA4H P09960 1/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31194858 0.92 MAPK13 (0.54) MAPK13MAPK12MAPK11MAPK14PTGS2
SCHEMBL29154641 0.86 MAPK13 (0.65) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL6539871 0.85 ESR2 (0.53) ESR2NOX1ESR1MAPTTP53
SCHEMBL6231069 0.84 ESR2 (0.51) ESR2NOX1ESR1MAPTTP53
SCHEMBL13772755 0.83 MAPK13 (0.69) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL3276327 0.81 MAPK14 (0.71) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL6208355 0.81 ESR2 (0.49) ESR2NOX1ESR1MAPTTP53
SCHEMBL6233898 0.81 ESR2 (0.49) ESR2NOX1ESR1MAPTTP53
SCHEMBL6538831 0.80 ESR2 (0.47) ESR2NOX1ESR1MAPTTP53
SCHEMBL6230071 0.80 ESR2 (0.47) ESR2NOX1ESR1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583749-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE Astellas Pharma Inc. (JP) 2005-10-12 EP disclosed
WO-2004065374-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE ASTELLAS PHARMA INC. (JP) 2004-08-05 WO disclosed