SCHEMBL6231276

SCHEMBL6231276

[c]1ccc2c(c1)ccn2COCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
CDK4 P11802 4/20 0.34
CCND1 P24385 4/20 0.34
ADORA2A P29274 1/20 0.34
KMT2A Q03164 1/20 0.33
APP P05067 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK14 Q16539 3/20 0.31
HTR6 P50406 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
AGER Q15109 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028017 0.80 HTR6 (0.49) CDK4CCND1KMT2AAPPHTR6
SCHEMBL16720003 0.78 CDK4 (0.44) CDK4CCND1KMT2AHSD17B10
SCHEMBL6231638 0.75 HTR2C (0.33) CDK4CCND1
SCHEMBL16719749 0.72 CYP3A4 (0.45) TSHRALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5068779 0.71 PLA2G4A (0.44) KMT2A
SCHEMBL6228700 0.70 CDK4 (0.35) CDK4CCND1KMT2A
SCHEMBL189124 0.70 CDK4 (0.35) CDK4CCND1KMT2A
Phosphoric Acid SCHEMBL27354178 0.69 KDM4E (0.37) TSHRKMT2AAPPHSD17B10ALDH1A1
SCHEMBL3200268 0.68 HTR6 (0.49) CDK4CCND1KMT2AAPPHTR6
SCHEMBL1660960 0.68 KMT2A (0.60) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1595866-B1 Cyanopyrrolidines useful for the treatment of inter alia metabolic syndrome SANWA KAGAKU KENKYUSHO CO (JP) 2016-06-08 EP disclosed
EP-1595866-A1 COMPOUND INHIBITING DIPEPTIDYL PEPTIDASE IV Sanwa Kagaku Kenkyusho Co., Ltd. (JP) 2005-11-16 EP disclosed