SCHEMBL6232312

SCHEMBL6232312

COc1ccc2[nH]c3cc(-c4ccc([N+](=O)[O-])cc4Br)c4c(c3c2c1)C(=O)NC4=O

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
WEE1 P30291 13/20 0.59
CHEK1 O14757 11/20 0.59
CTSV O60911 1/20 0.55
CTSL P07711 1/20 0.55
PDGFRB P09619 1/20 0.52
ROCK2 O75116 2/20 0.47
CCNB2 O95067 2/20 0.46
CDK1 P06493 2/20 0.46
CCNB1 P14635 2/20 0.46
GSK3B P49841 2/20 0.46
CDK5 Q00535 2/20 0.46
CDK5R1 Q15078 2/20 0.46
CCNB3 Q8WWL7 2/20 0.46
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5828397 0.89 WEE1 (0.70) WEE1CHEK1CTSVCTSLPDGFRB
SCHEMBL5828032 0.86 WEE1 (0.70) WEE1CHEK1CTSVCTSLPDGFRB
SCHEMBL5829115 0.85 WEE1 (0.71) WEE1CHEK1GSK3BCDK5CDK2
SCHEMBL5827617 0.83 WEE1 (0.74) WEE1CHEK1CTSVCTSLPDGFRB
SCHEMBL5827976 0.83 WEE1 (0.77) WEE1CHEK1PDGFRBROCK2GSK3B
SCHEMBL5829332 0.81 WEE1 (0.73) WEE1CHEK1PDGFRBROCK2
SCHEMBL5829421 0.79 WEE1 (0.70) WEE1CHEK1PDGFRBROCK2CCNE1
SCHEMBL5828572 0.79 WEE1 (0.72) WEE1CHEK1
SCHEMBL5828726 0.78 WEE1 (0.83) WEE1CHEK1PDGFRBROCK2GSK3B
SCHEMBL5829311 0.78 CTSV (0.58) WEE1CHEK1CTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501831-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2005-02-02 EP disclosed
WO-2003091255-A1 INHIBITORS OF CHECKPOINT KINASES (WEE1 AND CHK1) WARNER-LAMBERT COMPANY LLC (US) 2003-11-06 WO disclosed