SCHEMBL6232600

SCHEMBL6232600

CCC#CCOc1cc(N)c(Cl)cc1C(=O)NC1C2CCC1CN(Cc1ccccc1)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.56
DRD2 P14416 6/20 0.55
DRD3 P35462 5/20 0.55
HTR3A P46098 3/20 0.55
CYP3A4 P08684 2/20 0.55
ADRA2A P08913 2/20 0.55
ADRA2B P18089 2/20 0.55
ADRA2C P18825 2/20 0.55
HTR2A P28223 2/20 0.55
HTR2C P28335 2/20 0.55
HTR2B P41595 2/20 0.55
ACHE P22303 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
SLC6A2 P23975 1/20 0.55
ADRA1A P35348 1/20 0.55
OPRK1 P41145 1/20 0.55
CHRNA4 P43681 1/20 0.55
SLC6A3 Q01959 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6236267 0.99 DRD4 (0.55) DRD4DRD2DRD3HTR3ACYP3A4
SCHEMBL6234223 0.87 ADRA2A (0.50) HTR3AADRA2AADRA2BADRA2CHTR2A
Hydrochloric Acid SCHEMBL6232454 0.86 ADRA2A (0.49) HTR3AADRA2AADRA2BADRA2CHTR2A
SCHEMBL7243555 0.86 DRD4 (0.73) DRD4DRD2DRD3HTR3ACYP3A4
SCHEMBL6266458 0.84 ADRA2A (0.48) HTR3AADRA2AADRA2BADRA2CHTR2A
Hydrochloric Acid SCHEMBL6268711 0.84 ADRA2A (0.47) HTR3AADRA2AADRA2BADRA2CHTR2A
Hydrochloric Acid SCHEMBL6237211 0.82 ADRA2A (0.51) HTR3AADRA2AADRA2BADRA2CHTR2A
SCHEMBL4888712 0.81 DRD4 (0.55) DRD4DRD2DRD3HTR3ACYP3A4
SCHEMBL4888708 0.81 DRD4 (0.55) DRD4DRD2DRD3HTR3ACYP3A4
SCHEMBL6238770 0.81 ADRA2A (0.49) HTR3AADRA2AADRA2BADRA2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007600-A2 NOVEL METHODS USING AMINOBENZOIC ACID COMPOUNDS EISAI CO., LTD. (JP) 2005-01-27 WO disclosed