SCHEMBL6232613

SCHEMBL6232613

CCCC(NC(=O)c1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 7/20 0.44
TAS1R1 Q7RTX1 7/20 0.44
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
TSHR P16473 3/20 0.40
CTSK P43235 2/20 0.39
MAPK1 P28482 1/20 0.38
PSMD14 O00487 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HPGD P15428 1/20 0.37
PKM P14618 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ROCK2 O75116 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043124 0.90 POLB (0.34) TAS1R3TAS1R1NPC1RAB9ATSHR
SCHEMBL4043857 0.88 CTSK (0.44) CTSK
SCHEMBL4041145 0.87 CTSK (0.45) NPC1RAB9ATSHRCTSKMAPK1
SCHEMBL4040234 0.87 CTSK (0.54) NPC1RAB9ACTSKALDH1A1LMNA
SCHEMBL4039055 0.86 CTSK (0.54) RAB9ACTSKALDH1A1
SCHEMBL4041463 0.86 CTSK (0.43) TAS1R3TAS1R1RAB9ACTSKKMT2A
SCHEMBL4041112 0.86 CTSK (0.46) CTSK
SCHEMBL4040030 0.86 CTSK (0.41) NPC1RAB9ACTSKSMN1; SMN2
SCHEMBL4040328 0.85 CTSK (0.42) TAS1R3TAS1R1CTSK
SCHEMBL4045200 0.85 CTSK (0.45) NPC1RAB9ACTSKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed