SCHEMBL6232632

SCHEMBL6232632

NC(=O)c1ccc(Cl)c(COc2cnccn2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 3/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SGMS2 Q8NHU3 2/20 0.38
HTR2A P28223 1/20 0.38
KCNH2 Q12809 1/20 0.38
MAPT P10636 2/20 0.37
AGTR1 P30556 1/20 0.37
RXRA P19793 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37
SIRT1 Q96EB6 1/20 0.37
SIRT3 Q9NTG7 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079221 0.85 MAOB (0.45) HTR1ASMN1; SMN2RXRAGRIN1GRIN2B
SCHEMBL6079731 0.80 RXRA (0.40) SLC6A4SLC6A2SLC6A3SGMS2RXRA
SCHEMBL6078807 0.76 RAB9A (0.51) SGMS2
SCHEMBL6242298 0.73 RAB9A (0.46) SGMS2
SCHEMBL18339340 0.70 KCNH2 (0.38) SGMS2KCNH2
SCHEMBL2892451 0.69 SLC6A4 (0.50) KMT2ASLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL27722152 0.69 SLC6A4 (0.50) KMT2AHTR1ASLC6A4SLC6A2SLC6A3
SCHEMBL38662084 0.67 HDAC8 (0.61) SLC6A4HTR2AKCNH2
SCHEMBL5860852 0.66 TSHR (0.47) KMT2ASMN1; SMN2KDM4E
SCHEMBL6080064 0.66 MAOB (0.53) KMT2AHTR1ASMN1; SMN2SIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005002673-A1 RAF KINASE INHIBITORS ASTEX THERAPEUTICS LIMITED (GB) 2005-01-13 WO disclosed