SCHEMBL6232785

SCHEMBL6232785

NC1(c2cccc(C(F)(F)F)c2)N=CC=CN1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.43
SLC6A4 P31645 3/20 0.40
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A3 Q01959 2/20 0.35
SLC6A2 P23975 1/20 0.35
PNMT P11086 1/20 0.34
KCNN4 O15554 2/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
IDO1 P14902 2/20 0.33
IKBKB O14920 1/20 0.33
TDO2 P48775 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1172321 0.77 KDM1A (0.43) KDM1ASLC6A4TSHRMAPK1SLC6A3
SCHEMBL10763454 0.76 MAOA (0.33) KDM1APNMTBACE1BACE2
SCHEMBL3107125 0.70 KDM1A (0.42) KDM1ASLC6A4TSHRMAPK1SLC6A3
SCHEMBL7104862 0.69 MAPT (0.36) SLC6A4SLC6A3SLC6A2
SCHEMBL16014198 0.69 KDM1A (0.43) KDM1ASLC6A4TSHRMAPK1SLC6A3
SCHEMBL1391271 0.68 DHFR (0.43) KDM1ASLC6A4TSHRMAPK1BACE1
SCHEMBL22369879 0.67 KDM1A (0.56) KDM1ASLC6A4TSHRMAPK1SLC6A3
SCHEMBL1420518 0.66 KDM1A (0.59) KDM1ASLC6A4TSHRMAPK1SLC6A3
Hydrochloric Acid SCHEMBL20564061 0.66 KDM1A (0.54) KDM1ASLC6A4TSHRMAPK1SLC6A3
Hydrochloric Acid SCHEMBL3001569 0.65 KDM1A (0.57) KDM1ASLC6A4TSHRMAPK1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed