SCHEMBL6232857

SCHEMBL6232857

Cn1c(CBr)cc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.56
MAPT P10636 9/20 0.47
GLS O94925 1/20 0.45
CYP1A2 P05177 1/20 0.43
ALDH1A1 P00352 5/20 0.42
PKM P14618 1/20 0.42
MEN1 O00255 5/20 0.42
KMT2A Q03164 5/20 0.42
RXFP1 Q9HBX9 1/20 0.42
LMNA P02545 5/20 0.41
CYP2D6 P10635 1/20 0.41
F2RL3 Q96RI0 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
F2R P25116 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP3A4 P08684 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HPGD P15428 1/20 0.40
KDM4E B2RXH2 1/20 0.39
APOBEC3A P31941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6230356 0.85 CYP19A1 (0.59) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL9486251 0.81 CYP19A1 (0.52) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL23320466 0.80 CYP19A1 (0.60) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL6233158 0.79 ALDH1A1 (0.61) CYP19A1MAPTALDH1A1PKMMEN1
SCHEMBL3481105 0.78 CYP19A1 (0.61) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL31036289 0.78 CYP19A1 (0.61) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL21774736 0.76 CYP19A1 (0.56) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL8032940 0.75 KCNJ1 (0.48) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL6637649 0.74 KCNJ1 (0.53) CYP19A1MAPTGLSCYP1A2ALDH1A1
SCHEMBL29540854 0.74 MAPT (0.43) CYP19A1MAPTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed