SCHEMBL8032940

SCHEMBL8032940

Cn1c(Cc2ccc(C#N)cc2)cc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 2/20 0.48
KCNH2 Q12809 2/20 0.48
CYP19A1 P11511 1/20 0.46
MAPT P10636 4/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
IDH1 O75874 1/20 0.40
DCTPP1 Q9H773 1/20 0.39
CYP1A2 P05177 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
CNR2 P34972 1/20 0.38
RORC P51449 1/20 0.38
F2RL3 Q96RI0 1/20 0.38
OPRM1 P35372 1/20 0.38
GLS O94925 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6637649 0.89 KCNJ1 (0.53) KCNJ1KCNH2CYP19A1MAPTALDH1A1
SCHEMBL8029974 0.79 ALDH1A1 (0.55) KCNJ1KCNH2MAPTALDH1A1MEN1
SCHEMBL8016775 0.79 BRPF1 (0.41) KCNJ1KCNH2KMT2AIDH1RORC
SCHEMBL8029881 0.77 KCNJ1 (0.46) KCNJ1KCNH2CYP19A1MAPTALDH1A1
SCHEMBL8030047 0.77 KMT2A (0.46) KMT2AIDH1
SCHEMBL7981313 0.77 ALDH1A1 (0.44) KCNJ1KCNH2MAPTALDH1A1GAA
SCHEMBL6230356 0.75 CYP19A1 (0.59) CYP19A1MAPTALDH1A1KDM4EMEN1
SCHEMBL6232857 0.75 CYP19A1 (0.56) CYP19A1MAPTALDH1A1KDM4EMEN1
SCHEMBL7360923 0.74 KCNJ1 (0.52) KCNJ1KCNH2CYP19A1RORC
SCHEMBL6159759 0.74 KMT2A (0.58) KCNJ1KCNH2CYP19A1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060166-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS Boehringer Ingelheim Pharma KG (DE) 2000-12-20 EP disclosed
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed
WO-1999040072-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-08-12 WO disclosed