SCHEMBL6233054

SCHEMBL6233054

COc1cc(CC#Cc2ccc3[nH]cc(CCc4ccc(C(=O)O)cc4)c(=O)c3c2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.43
MMP13 P45452 6/20 0.42
HAO1 Q9UJM8 2/20 0.37
SLC22A8 Q8TCC7 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ACACB O00763 2/20 0.35
HTR7 P34969 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.34
SLC13A5 Q86YT5 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
HTR1A P08908 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6260796 0.77 MMP13 (0.44) FFAR1MMP13SLC22A8ACACBLOXL2
SCHEMBL6297941 0.73 MMP13 (0.78) MMP13SLC22A8
SCHEMBL6231783 0.69 MMP13 (0.53) MMP13LOXL2
SCHEMBL6254579 0.67 MMP13 (0.40) FFAR1MMP13SLC22A8ACACBLOXL2
SCHEMBL6450474 0.66 MMP13 (0.36) MMP13SLC22A8
SCHEMBL6296011 0.64 MMP13 (0.69) MMP13SLC22A8
SCHEMBL6842418 0.64 FFAR1 (0.39) FFAR1MMP13
SCHEMBL6250624 0.64 MMP13 (0.38) FFAR1MMP13ACACBLOXL2
SCHEMBL6233684 0.64 MMP13 (0.49) MMP13SLC22A8
SCHEMBL6231728 0.64 MMP13 (0.49) MMP13SLC22A8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1525030-A1 COMBINATION OF AN ALLOSTERIC ALKYNE INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-04-27 EP disclosed
WO-2004007025-A1 COMBINATION OF AN ALLOSTERIC ALKYNE INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 THAT IS NOT CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed