SCHEMBL6450474

SCHEMBL6450474

COc1cc(CC#Cc2c(Cc3ccc(C(=O)O)cc3)c(=O)c3ccccc3n2C)ccn1.O=c1cc[nH]c2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 7/20 0.36
SLC22A8 Q8TCC7 1/20 0.36
MAPK8 P45983 3/20 0.32
MAPK9 P45984 1/20 0.32
PTGER4 P35408 2/20 0.32
RHEB Q15382 1/20 0.31
POLB P06746 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
PPARG P37231 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
PTPN5 P54829 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6853866 0.74 MMP13 (0.44) MMP13SLC22A8PTGER4POLBKDM4E
SCHEMBL6266827 0.74 MMP13 (0.45) MMP13SLC22A8MAPK8MAPK9PTGER4
SCHEMBL6260796 0.67 MMP13 (0.44) MMP13SLC22A8
SCHEMBL6233054 0.66 FFAR1 (0.43) MMP13SLC22A8
SCHEMBL7035431 0.64 MMP13 (0.48) MMP13SLC22A8MEN1ALDH1A1KMT2A
SCHEMBL6231783 0.64 MMP13 (0.53) MMP13
SCHEMBL6297941 0.62 MMP13 (0.78) MMP13SLC22A8
SCHEMBL6296011 0.62 MMP13 (0.69) MMP13SLC22A8
SCHEMBL6250624 0.62 MMP13 (0.38) MMP13ALDH1A1
SCHEMBL6233684 0.62 MMP13 (0.49) MMP13SLC22A8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1536786-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2005-06-08 EP disclosed
WO-2004006913-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed