SCHEMBL6233535

SCHEMBL6233535

COc1ccc2c(Cc3ccc(OCCC4CCCCN4)cc3)c(-c3ccc(S(C)(=O)=O)cc3)ccc2c1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.56
ESR2 Q92731 4/20 0.56
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.40
CHEK2 O96017 1/20 0.39
SSTR2 P30874 4/20 0.38
LTA4H P09960 6/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6234142 0.91 ESR1 (0.70) ESR1ESR2CHEK2SSTR2LTA4H
SCHEMBL6234450 0.85 CHEK2 (0.46) ESR1ESR2PTGS2PTGS1CHEK2
SCHEMBL6238825 0.83 ESR1 (0.42) ESR1ESR2PTGS2CHEK2SSTR2
SCHEMBL3115469 0.82 ESR1 (0.81) ESR1ESR2LTA4H
SCHEMBL3714380 0.81 ESR1 (0.64) ESR1ESR2CHEK2SSTR2LTA4H
Hydrochloric Acid SCHEMBL5256714 0.81 ESR1 (0.66) ESR1ESR2CHEK2SSTR2LTA4H
SCHEMBL1359104 0.79 LTA4H (0.39) ESR1ESR2CHEK2LTA4H
SCHEMBL6136215 0.79 ESR1 (0.65) ESR1ESR2CHEK2SSTR2LTA4H
SCHEMBL6148234 0.78 ESR1 (0.69) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6004702 0.78 ESR1 (0.59) ESR1ESR2CHEK2SSTR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530470-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP ELI LILLY AND COMPANY (US) 2005-05-18 EP disclosed
WO-2004009086-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP ELI LILLY AND COMPANY (US) 2004-01-29 WO disclosed