SCHEMBL6238825

SCHEMBL6238825

COc1ccc2c(C(O)c3ccc(OCCC4CCCCN4)cc3)c(-c3ccc(S(C)(=O)=O)cc3)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.42
ESR2 Q92731 6/20 0.42
CHEK2 O96017 1/20 0.40
PTGS2 P35354 1/20 0.39
SSTR2 P30874 7/20 0.38
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205268 0.85 SSTR2 (0.39) CHEK2SSTR2
SCHEMBL6234450 0.84 CHEK2 (0.46) ESR1ESR2CHEK2PTGS2SSTR2
SCHEMBL6233535 0.83 ESR1 (0.56) ESR1ESR2CHEK2PTGS2SSTR2
SCHEMBL6205481 0.83 SSTR2 (0.39) CHEK2SSTR2
SCHEMBL3107296 0.83 ESR1 (0.62) ESR1ESR2
SCHEMBL5706983 0.79 MAPK1 (0.38) SSTR2
SCHEMBL5707024 0.78 SSTR2 (0.37) SSTR2
SCHEMBL6148234 0.78 ESR1 (0.69) ESR1ESR2CHEK2SSTR2
SCHEMBL6236259 0.77 ESR1 (0.53) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6111606 0.77 ESR1 (0.69) ESR1ESR2CHEK2SSTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530470-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP ELI LILLY AND COMPANY (US) 2005-05-18 EP disclosed
WO-2004009086-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS CONTAINING A PHENYLSULFONYL GROUP ELI LILLY AND COMPANY (US) 2004-01-29 WO disclosed