SCHEMBL6234576

SCHEMBL6234576

COc1ccc(CC#N)c(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.45
POLB P06746 1/20 0.45
CYP1A2 P05177 1/20 0.45
CHRM2 P08172 1/20 0.45
SLC6A4 P31645 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
KDM4E B2RXH2 6/20 0.44
TSHR P16473 1/20 0.44
APOBEC3A P31941 1/20 0.44
CTDSP1 Q9GZU7 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
ALDH1A1 P00352 4/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9786028 0.85 AOC3 (0.39) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL10648349 0.85 AOC3 (0.39) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL6356440 0.84 AOC3 (0.38) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL150075 0.84 CA1 (0.40) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL4160051 0.83 SMN1; SMN2 (0.46) SMN1; SMN2POLBCYP1A2KDM4ETSHR
SCHEMBL7273837 0.82 SLC2A1 (0.42) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL8248932 0.82 BCHE (0.48) SMN1; SMN2POLBKDM4ETSHRMAPT
SCHEMBL28771054 0.81 AOC3 (0.36) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL7274049 0.81 AOC3 (0.36) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL954640 0.81 MEN1 (0.47) POLBKDM4ETSHRALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed
US-20070142399-A1 Dual function drugs and uses thereof PSYCHIATRIC GENOMICS, INC. (US) 2007-06-21 US disclosed
US-20070142399-A1 Dual function drugs and uses thereof PSYCHIATRIC GENOMICS, INC. (US) 2007-06-21 US disclosed
EP-1066227-B1 PROCESS OF PREPARING DISCOTIC LIQUID CRYSTALLINE COMPOUNDS MERCK PATENT GMBH (DE) 2005-12-28 EP disclosed
EP-1523556-A1 METHODS OF TREATING CONDITIONS ASSOCIATED WITH AN EDG-1 RECEPTOR SRI INTERNATIONAL (US) 2005-04-20 EP disclosed
WO-2004009816-A1 METHODS OF TREATING CONDITIONS ASSOCIATED WITH AN EDG-1 RECEPTOR CERETEK LLC (US) 2004-01-29 WO disclosed
US-6534135-B1 Process of preparing discotic liquid crystalline compounds MERCK PATENT GESELLSCHAFT (DE) 2003-03-18 US disclosed
EP-1066227-A1 PROCESS OF PREPARING DISCOTIC LIQUID CRYSTALLINE COMPOUNDS MERCK PATENT GmbH (DE) 2001-01-10 EP disclosed
EP-0957092-A1 Ring-closed dihydropyridines and their use in the preparation of pharmaceutical compositions Boehringer Ingelheim Pharma KG (DE) 1999-11-17 EP disclosed
WO-1999048844-A1 PROCESS OF PREPARING DISCOTIC LIQUID CRYSTALLINE COMPOUNDS MERCK PATENT GMBH (DE) 1999-09-30 WO disclosed
US-5861412-A CARDIOPROTECTIVE AGENTS, CEREBROPROTECTIVE AGENTS, AGENTS FOR TREATING CHRONIC INFLAMMATORY PROCESSES, ANTIPROLIFERATIVE AGENTS AND AS AGENTS FOR TREATING ULCERATIVE COLITIS AND CROHN'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1999-01-19 US disclosed
US-5674878-A ANTIPROLIFERATIVE,-TUMOR AND -CARCINOGENIC AGENTS; ULCERATIVE COLITIS; CROHN*S DISEASE BOEHRINGER INGELHEIM KG (DE) 1997-10-07 US disclosed
US-5643919-A TREATMENT OF CROHN*S DISEASE, ULCERATIVE COLITIS BOEHRINGER INGELHEIM KG (DE) 1997-07-01 US disclosed
WO-1994000435-A1 RING-CLOSED DIHYDROPYRIDINES AND THEIR USE IN THE PREPARATION OF PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM KG (DE) 1994-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070142399-A1 Dual function drugs and uses thereof COMT, DRD2, SLC6A3 AOC3 943/4885SMN1; SMN2 4424/4885POLB 3939/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.