SCHEMBL6234869

SCHEMBL6234869

CN(C)CCN1CCN(CCCOc2ccc(-c3cnc4nc(-c5cccs5)c(-c5cccs5)nc4c3)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.48
KCNH2 Q12809 1/20 0.48
HRH1 P35367 2/20 0.46
HRH2 P25021 1/20 0.46
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
DRD3 P35462 2/20 0.40
MAPK1 P28482 1/20 0.40
CXCR1 P25024 2/20 0.39
HTR3A P46098 3/20 0.39
HRH4 Q9H3N8 1/20 0.38
TLR9 Q9NR96 1/20 0.37
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235648 0.90 HRH3 (0.51) HRH3KCNH2HRH1HRH2RAB9A
SCHEMBL6255922 0.87 HRH3 (0.51) HRH3KCNH2HRH1HRH2RAB9A
SCHEMBL6240919 0.80 RPS6KB2 (0.44) HRH3KCNH2RAB9ANPC1MAPK1
SCHEMBL6233813 0.80 RPS6KB2 (0.43) HRH3KCNH2RAB9ANPC1MAPK1
SCHEMBL6237806 0.80 CHEK2 (0.40) CXCR1
SCHEMBL6237136 0.79 RPS6KB2 (0.44) RAB9ANPC1MAPK1
SCHEMBL6233986 0.73 ACP1 (0.39) HRH3KCNH2
SCHEMBL6234523 0.72 CYP1A2 (0.42) MAPK1
SCHEMBL6240032 0.72 RPS6KB2 (0.42) HRH3KCNH2RAB9ANPC1MAPK1
SCHEMBL6236199 0.71 RPS6KB2 (0.41) HRH3KCNH2RAB9ANPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007099-A2 PKB INHIBITORS AS ANTI-TUMOR AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-27 WO disclosed