SCHEMBL6233986

SCHEMBL6233986

c1csc(-c2nc3cc(-c4ccc(OCCCC5CCNC5)cc4)cnc3nc2-c2cccs2)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.39
ROCK1 Q13464 1/20 0.37
PRKCZ Q05513 2/20 0.37
CHEK1 O14757 1/20 0.36
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 1/20 0.36
HDAC3 O15379 3/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC2 Q92769 3/20 0.35
RPS6KB2 Q9UBS0 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
KCNH2 Q12809 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
PBK Q96KB5 2/20 0.33
CHEK2 O96017 1/20 0.33
NPY1R P25929 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6233813 0.81 RPS6KB2 (0.43) RPS6KB2HRH3KCNH2
SCHEMBL6240919 0.79 RPS6KB2 (0.44) RPS6KB2HRH3KCNH2
SCHEMBL6237136 0.78 RPS6KB2 (0.44) RPS6KB2CHEK2
SCHEMBL6255922 0.75 HRH3 (0.51) SLC6A4HRH3KCNH2
SCHEMBL6235648 0.75 HRH3 (0.51) HRH3KCNH2
SCHEMBL6234869 0.73 HRH3 (0.48) HRH3KCNH2
SCHEMBL6240032 0.72 RPS6KB2 (0.42) RPS6KB2HRH3KCNH2
SCHEMBL6236199 0.71 RPS6KB2 (0.41) RPS6KB2HRH3KCNH2
SCHEMBL6237798 0.71 RPS6KB2 (0.52) RPS6KB2
SCHEMBL6237105 0.71 RPS6KB2 (0.49) RPS6KB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005007099-A2 PKB INHIBITORS AS ANTI-TUMOR AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-27 WO disclosed