SCHEMBL6234890

SCHEMBL6234890

CS(=O)(=O)c1ccc(-c2nnc(-c3ccccc3NCC3=CCOO3)[nH]2)cc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.38
SCD O00767 2/20 0.35
FADS1 O60427 1/20 0.35
WNT3A P56704 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
JAK2 O60674 1/20 0.33
PTK2 Q05397 1/20 0.33
CNR1 P21554 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6234886 0.82 PTGS2 (0.38) PTGS2SCDFADS1WNT3ATNKS2
SCHEMBL13605666 0.79 PTGS2 (0.48) PTGS2JAK2PTK2CNR1KDR
SCHEMBL4178035 0.76 PDE5A (0.48) PTGS2KDR
SCHEMBL4182630 0.74 BRD4 (0.46) PTGS2SCDFADS1WNT3ATNKS2
SCHEMBL6234875 0.69 EED (0.38) PTGS2SCDFADS1WNT3ATNKS2
SCHEMBL4176801 0.65 EED (0.52) PTGS2KDR
SCHEMBL4181032 0.64 KDR (0.58) KDR
SCHEMBL4174127 0.64 KDR (0.74) PTGS2SCDWNT3ATNKS2KDR
SCHEMBL4180618 0.64 PTGS2 (0.52) PTGS2KDR
SCHEMBL4179144 0.63 PTGS2 (0.49) PTGS2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005004818-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS ANTICANCER AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-20 WO disclosed