SCHEMBL6234886

SCHEMBL6234886

CS(=O)(=O)c1ccc(-c2nnc(-c3ccccc3NCC3=COCO3)[nH]2)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.38
SCD O00767 2/20 0.35
FADS1 O60427 1/20 0.35
PTGS1 P23219 1/20 0.34
EED O75530 1/20 0.34
SUZ12 Q15022 1/20 0.34
EZH2 Q15910 1/20 0.34
WNT3A P56704 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
JAK2 O60674 1/20 0.33
PTK2 Q05397 1/20 0.33
CNR1 P21554 1/20 0.33
KDR P35968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6234890 0.82 PTGS2 (0.38) PTGS2SCDFADS1WNT3ATNKS2
SCHEMBL4178035 0.80 PDE5A (0.48) PTGS2PTGS1KDR
SCHEMBL13605666 0.79 PTGS2 (0.48) PTGS2PTGS1JAK2PTK2CNR1
SCHEMBL4178043 0.77 PTGS2 (0.38) PTGS2SCDFADS1PTGS1
SCHEMBL4173252 0.74 PTGS2 (0.37) PTGS2PTGS1
SCHEMBL6234882 0.74 PTGS2 (0.36) PTGS2SCDFADS1PTGS1WNT3A
SCHEMBL4182630 0.74 BRD4 (0.46) PTGS2SCDFADS1PTGS1WNT3A
SCHEMBL6234875 0.69 EED (0.38) PTGS2SCDFADS1PTGS1EED
SCHEMBL4173244 0.67 PDE5A (0.52) KDR
SCHEMBL4182621 0.65 TUBB4A (0.50) PTGS2EEDSUZ12EZH2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005004818-A2 HETEROCYCLIC COMPOUNDS AND THEIR USE AS ANTICANCER AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2005-01-20 WO disclosed