SCHEMBL6235042

SCHEMBL6235042

O=C(OCc1ccc(F)c(F)c1)N1CCOCC1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.62
KMT2A Q03164 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
GRIN2B Q13224 1/20 0.49
NPC1 O15118 1/20 0.47
TSHR P16473 4/20 0.46
BCL9 O00512 1/20 0.45
CTNNB1 P35222 1/20 0.45
AOC3 Q16853 2/20 0.44
PRKDC P78527 1/20 0.44
MAPT P10636 1/20 0.43
RECQL P46063 1/20 0.43
TP53 P04637 1/20 0.43
GPR183 P32249 1/20 0.43
ENPP2 Q13822 1/20 0.43
ATXN2 Q99700 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235843 0.86 MEN1 (0.55) MEN1KMT2ANPSR1GRIN2BTSHR
SCHEMBL4678059 0.83 DPP4 (0.55) MEN1KMT2ANPSR1GRIN2BNPC1
Hydrochloric Acid SCHEMBL4680856 0.82 DPP4 (0.54) MEN1KMT2ANPSR1GRIN2BNPC1
SCHEMBL6236015 0.78 MEN1 (0.62) MEN1KMT2ANPSR1TSHRENPP2
SCHEMBL1337663 0.78 KMT2A (0.97) MEN1KMT2ANPSR1GRIN2BNPC1
SCHEMBL14095609 0.78 KMT2A (0.97) MEN1KMT2ANPSR1GRIN2BNPC1
SCHEMBL6235265 0.77 MEN1 (0.53) MEN1KMT2ANPSR1GRIN2BNPC1
SCHEMBL542951 0.77 ENPP2 (0.54) MEN1KMT2ANPSR1NPC1MAPT
SCHEMBL1314311 0.75 MEN1 (0.71) MEN1KMT2ANPSR1GRIN2BNPC1
Hydrochloric Acid SCHEMBL1313138 0.74 MEN1 (0.69) MEN1KMT2ANPSR1GRIN2BNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1390034-A4 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2005-07-13 EP disclosed
EP-1390034-A1 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2004-02-25 EP disclosed
WO-2002080928-A1 N-SUBSTITUTED NONARYL-HETEROCYCLO AMIDYL NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2002-10-17 WO disclosed