SCHEMBL6235301

SCHEMBL6235301

CNC(=O)Nc1ccc(-c2cccc(C(F)(F)F)c2)nc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.58
MAPT P10636 3/20 0.55
NPC1 O15118 1/20 0.55
PIK3CD O00329 1/20 0.53
PIK3CA P42336 1/20 0.53
PIK3CG P48736 1/20 0.53
FYN P06241 1/20 0.49
KDM1A O60341 2/20 0.49
MAOB P27338 2/20 0.49
PSEN1 P49768 1/20 0.48
PSEN2 P49810 1/20 0.48
APH1B Q8WW43 1/20 0.48
NCSTN Q92542 1/20 0.48
APH1A Q96BI3 1/20 0.48
PSENEN Q9NZ42 1/20 0.48
KCNQ3 O43525 1/20 0.48
KCNQ2 O43526 1/20 0.48
KCNE1 P15382 1/20 0.48
KCNQ1 P51787 1/20 0.48
KIF11 P52732 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6233041 0.88 FYN (0.62) DHODHMAPTNPC1PIK3CDPIK3CA
SCHEMBL6257855 0.85 DHODH (0.58) DHODHMAPTNPC1PIK3CDPIK3CA
SCHEMBL6235084 0.85 KIF11 (0.67) DHODHMAPTNPC1PIK3CDPIK3CA
SCHEMBL6235521 0.84 DHODH (0.57) DHODHMAPTNPC1PIK3CDPIK3CA
SCHEMBL6235785 0.84 TP53 (0.62) DHODHMAPTNPC1PIK3CDPIK3CA
SCHEMBL6239029 0.80 BAZ2B (0.64) DHODHNPC1PIK3CDPIK3CAPIK3CG
SCHEMBL6243512 0.77 DHODH (0.54) DHODHPIK3CDPIK3CAPIK3CGFYN
SCHEMBL2632866 0.77 MAPT (0.73) MAPTMAPK1MEN1KMT2AKDR
SCHEMBL6236761 0.76 DHODH (0.52) DHODHPIK3CDPIK3CAPIK3CGFYN
SCHEMBL5934519 0.75 TRPV1 (0.56) DHODHBRAFLCKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed