SCHEMBL6236041

SCHEMBL6236041

COc1ccccc1CS(=O)(=O)c1ccc(=O)[nH]n1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 18/20 0.69
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
AR P10275 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238316 0.83 AKR1B1 (0.53) AKR1B1
SCHEMBL6238212 0.82 AKR1B1 (1.00) AKR1B1
SCHEMBL6207787 0.76 AKR1B1 (0.62) AKR1B1
SCHEMBL6235231 0.76 AKR1B1 (1.00) AKR1B1AR
SCHEMBL6238246 0.75 AKR1B1 (0.76) AKR1B1
SCHEMBL6234461 0.75 AKR1B1 (0.76) AKR1B1
SCHEMBL7276901 0.74 AR (0.55) PTGS1PTGS2AR
SCHEMBL6237022 0.71 AKR1B1 (0.76) AKR1B1
SCHEMBL2719015 0.70 HTT (0.53)
SCHEMBL6238324 0.70 AKR1B1 (1.00) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236720-B1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors PFIZER PROD INC (US) 2005-06-15 EP claimed
US-6730674-B2 ANTIDIABETIC AGENTS PFIZER INC 2004-05-04 US claimed
US-20030004139-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors MARTIN WILLIAM H (US) 2003-01-02 US claimed
EP-1236720-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors Pfizer Products Inc. (US) 2002-09-04 EP claimed
EP-1236720-B1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors PFIZER PROD INC (US) 2005-06-15 EP disclosed
US-6730674-B2 ANTIDIABETIC AGENTS PFIZER INC 2004-05-04 US disclosed
US-20030004139-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors MARTIN WILLIAM H (US) 2003-01-02 US disclosed
EP-1236720-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors Pfizer Products Inc. (US) 2002-09-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030004139-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors ALDOA, PDXK, AKR1B1 AKR1B1 3/4885PTGS1 1328/4885PTGS2 1342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.