SCHEMBL6238316

SCHEMBL6238316

COc1ccc(OC)c(CS(=O)(=O)c2ccc(=O)[nH]n2)c1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 14/20 0.53
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
LMNA P02545 1/20 0.42
HSD17B10 Q99714 1/20 0.42
POLB P06746 1/20 0.41
ADRA1A P35348 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236041 0.83 AKR1B1 (0.69) AKR1B1
SCHEMBL6240241 0.80 AKR1B1 (0.58) AKR1B1PDE4APDE4BPDE4CPDE4D
SCHEMBL29594234 0.70 IDO1 (0.57) HSD17B10ADRA1ATAAR1IDO1
SCHEMBL6207869 0.70 AKR1B1 (1.00) AKR1B1LMNAPOLB
SCHEMBL8480289 0.69 LMNA (0.60) AKR1B1PDE4APDE4BPDE4CPDE4D
SCHEMBL6237022 0.69 AKR1B1 (0.76) AKR1B1
SCHEMBL6239197 0.68 AKR1B1 (0.62) AKR1B1
SCHEMBL6238212 0.68 AKR1B1 (1.00) AKR1B1
SCHEMBL6241896 0.68 AKR1B1 (1.00) AKR1B1
SCHEMBL6234479 0.67 AKR1B1 (0.78) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1236720-B1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors PFIZER PROD INC (US) 2005-06-15 EP disclosed
US-6730674-B2 ANTIDIABETIC AGENTS PFIZER INC 2004-05-04 US disclosed
US-20030004139-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors MARTIN WILLIAM H (US) 2003-01-02 US disclosed
EP-1236720-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors Pfizer Products Inc. (US) 2002-09-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030004139-A1 Sulfonyl pyridazinone compounds useful as aldose reductase inhibitors ALDOA, PDXK, AKR1B1 AKR1B1 3/4885PDE4A 1617/4885PDE4B 1528/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.