SCHEMBL6236434

SCHEMBL6236434

COC1NC(=O)N(C)C1=O

nearest known ligand 0.30

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232526 0.76 MAPT (0.33) GAA
SCHEMBL6231077 0.73 KDM4A (0.33)
SCHEMBL6238691 0.70 KDM4A (0.41) MEN1KMT2ATP53GAA
SCHEMBL145660 0.67
SCHEMBL12050006 0.67
SCHEMBL6232302 0.66 LMNA (0.47) KMT2AGAA
SCHEMBL10684022 0.65
SCHEMBL2726860 0.65
SCHEMBL14345533 0.65
SCHEMBL1361386 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0160618-A1 Hydantoin derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1985-11-06 EP claimed
EP-3639821-B1 CARCINOGENESIS INHIBITOR NAT CANCER CT (JP) 2024-08-28 EP disclosed
CN-110740729-B Carcinogenesis inhibitor 国立研究开发法人国立癌症研究中心 2023-05-16 CN disclosed
US-11464762-B2 Carcinogenesis inhibitor NATIONAL CANCER CENTER (JP) 2022-10-11 US disclosed
US-20200276163-A1 CARCINOGENESIS INHIBITOR NATIONAL CANCER CENTER (JP) 2020-09-03 US disclosed
EP-3639821-A1 CARCINOGENESIS INHIBITOR National Cancer Center (JP) 2020-04-22 EP disclosed
EP-1243261-B1 Use of a hydantoin derivative in a pharmaceutical composition against hypoalbuminaemia NIPPON ZOKI PHARMACEUTICAL CO (JP) 2005-04-27 EP disclosed
EP-1070706-B1 Process for the preparation of 1-substituted 5-hydroxy-imidazolin-2,4-diones and 1-substituted 5-alkoxy-imidazolin-2,4-diones BAYER CHEMICALS AG (DE) 2004-02-18 EP disclosed
EP-1018339-B1 Use of hydantoin derivatives for the preparation of a medicament for the treatment of intractable vasculitis. NIPPON ZOKI PHARMACEUTICAL CO (JP) 2003-05-02 EP disclosed
US-20020147228-A1 AGENT FOR HYPOALBUMINAEMIA NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2002-10-10 US disclosed
US-6365752-B1 REACTING GLYOXYLIC ACID AND AN N-SUBSTITUTED UREA IN AQUEOUS SOLUTION AND IN THE PRESENCE OF AN ACID CATALYST; EFFICIENCY; PURITY; NONTOXIC CHEMICAL INTERMEDIATES FOR DRUGS; INSECTICIDES; AMINO ACIDS AND TEXTILE ASSISTANTS BAYER AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed
US-6251929-B1 ADMINISTERING TO A PATIENT A HYDANTOIN DERIVATIVES AND SALTS AS THERAPEUTIC AND PREVENTIVE AGENTS FOR INTRACTABLE VASCULITIS SUCH AS MALIGNANT RHEUMATOID ARTHRITIS(MRA), PERIARTERITIS NODOSA, WEGENER'S GRANULOMATOSIS ETC. NIPPON ZOKI PHARMACEUTICALS CO., LTD. (JP) 2001-06-26 US disclosed
EP-0780125-B1 Use of hydantoin derivatives for the preparation of a medicament for the treatment of dieases associated with the presence of active oxygen and free radicals NIPPON ZOKI PHARMACEUTICAL CO (JP) 2001-04-18 EP disclosed
US-6197806-B1 USING A HYDANTOIN DERIVATIVE NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2001-03-06 US disclosed
EP-1070706-A1 Process for the preparation of 1-substituted 5-hydroxy-imidazolin-2,4-diones and 1-substituted 5-alkoxy-imidazolin-2,4-diones BAYER AG (DE) 2001-01-24 EP disclosed
EP-1018339-A1 Therapeutic agent for intractable vasculitis NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 2000-07-12 EP disclosed
EP-0780125-A2 Pharmaceutical composition containing a hydantoin derivative and use of said derivative NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-06-25 EP disclosed
EP-0160618-B1 HYDANTOIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1991-08-14 EP disclosed
US-4647574-A Hypoglycemic hydantoin derivatives NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1987-03-03 US disclosed
EP-0160618-A1 Hydantoin derivatives and pharmaceutical compositions containing them NIPPON ZOKI PHARMACEUTICAL CO. LTD. (JP) 1985-11-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11464762-B2 Carcinogenesis inhibitor APC, MKI67, HRAS MEN1 727/4885KMT2A 492/4885TP53 24/4885
US-20020147228-A1 AGENT FOR HYPOALBUMINAEMIA ALB, TTR, SERPINA6 MEN1 4444/4885KMT2A 4295/4885TP53 2399/4885
US-20200276163-A1 CARCINOGENESIS INHIBITOR APC, MKI67, HRAS MEN1 727/4885KMT2A 492/4885TP53 24/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.