SCHEMBL6236558

SCHEMBL6236558

CCCC(NC(=O)c1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 7/20 0.45
TAS1R1 Q7RTX1 7/20 0.45
CTSK P43235 2/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
TSHR P16473 2/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.39
GPR132 Q9UNW8 3/20 0.39
ROCK2 O75116 1/20 0.38
GFER P55789 1/20 0.38
HTRA1 Q92743 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046542 0.89 POLB (0.36) TAS1R3TAS1R1CTSKTSHRPKM
SCHEMBL4045236 0.88 CTSK (0.47) CTSKGPR132HTRA1
SCHEMBL4037490 0.86 CTSK (0.48) CTSKGPR132HTRA1NPC1RAB9A
SCHEMBL4037811 0.86 CTSK (0.57) CTSKGPR132HTRA1MEN1NPC1
SCHEMBL4039803 0.86 CTSK (0.49) CTSKGPR132
SCHEMBL4039065 0.86 CTSK (0.57) CTSKCHRNB2CHRNA7CHRNA4GPR132
SCHEMBL4039388 0.86 CTSK (0.45) CTSKCHRNB2CHRNA7CHRNA4GPR132
SCHEMBL4038068 0.85 CTSK (0.44) CTSKGPR132
SCHEMBL4038144 0.85 CTSK (0.45) TAS1R3TAS1R1CTSKGPR132HTRA1
SCHEMBL4042871 0.84 CTSK (0.48) CTSKGPR132HTRA1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed