SCHEMBL4046542

SCHEMBL4046542

CCCC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.36
BMP1 P13497 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
ESR2 Q92731 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TSHR P16473 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
EDNRA P25101 1/20 0.34
PKM P14618 1/20 0.34
CTSK P43235 2/20 0.33
MCHR1 Q99705 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
PAX8 Q06710 1/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050084 0.93 CTSK (0.41) POLBBMP1MEN1USP2ALDH1A1
SCHEMBL4043031 0.89 HTRA1 (0.37) CTSKPAX8ACACBGPR132
SCHEMBL6236558 0.89 TAS1R3 (0.45) MEN1KMT2ATSHRPKMCTSK
SCHEMBL4043650 0.88 BMP1 (0.36) POLBBMP1MEN1USP2ALDH1A1
SCHEMBL4047771 0.88 CTSK (0.39) CTSKACACBGPR132
SCHEMBL4044443 0.87 ALDH1A1 (0.38) ALDH1A1CTSKPAX8ACACBGPR132
SCHEMBL4040981 0.86 CTSK (0.35) ALDH1A1CTSKPAX8ACACBGPR132
SCHEMBL4050093 0.85 HTT (0.41) BMP1MEN1ALDH1A1MAPTKMT2A
SCHEMBL4045728 0.85 CTSK (0.35) ALDH1A1CTSKPAX8ACACBGPR132
SCHEMBL4041663 0.84 CTSK (0.35) MEN1USP2KMT2ATSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed