SCHEMBL6236885

SCHEMBL6236885

OCCc1ccc(Nc2nc[nH]c3ncc(-c4ccccc4)c2-3)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.55
ALK Q9UM73 1/20 0.55
CDK1 P06493 5/20 0.46
KDR P35968 5/20 0.46
MAPKAPK2 P49137 1/20 0.42
PDE4B Q07343 6/20 0.39
STAT6 P42226 1/20 0.39
MAPT P10636 3/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 2/20 0.37
GAA P10253 1/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677800 0.86 MAPT (0.46) CDC7ALKKDRMAPTMEN1
SCHEMBL6240412 0.83 ABCG2 (0.41) CDC7ALKCDK1KDRMAPT
SCHEMBL6270213 0.83 FGFR1 (0.44) KDRMAPTMEN1KMT2ALMNA
SCHEMBL6683647 0.83 PDE5A (0.41) KDRMAPTMEN1NPC1RAB9A
SCHEMBL6237608 0.81 CDC7 (0.35) CDC7ALKCDK1KDRMAPT
SCHEMBL6235443 0.80 TP53 (0.41) PDE4BMAPTNPC1RAB9AKMT2A
SCHEMBL6684324 0.76 MKNK1 (0.45) CDK1MAPTRAB9ATDP1MAPK1
SCHEMBL6881613 0.75 CDC7 (0.49) CDC7ALKCDK1KDRMAPKAPK2
SCHEMBL6876454 0.73 PTK2 (0.40) CDK1MAPTLMNAPIM1
SCHEMBL9986916 0.70 TNNI3K (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836613-B1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS METABASIS THERAPEUTICS INC (US) 2005-05-25 EP disclosed
EP-0836613-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-22 EP disclosed
WO-1996040707-A1 WATER-SOLUBLE ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed