SCHEMBL6237085

SCHEMBL6237085

Cn1c(C(F)(F)F)c(-c2ccc(C[C@H](N)C(=O)O)cc2)c(=O)n(C)c1=O

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 9/20 0.61
ITGA4 P13612 9/20 0.61
ITGB7 P26010 9/20 0.61
GRB2 P62993 1/20 0.46
PTPN1 P18031 2/20 0.43
SLC7A5 Q01650 2/20 0.43
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
TYR P14679 5/20 0.40
TPH1 P17752 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27511517 1.00 ITGB1 (0.61) ITGB1ITGA4ITGB7GRB2PTPN1
SCHEMBL5164910 0.88 ITGA4 (0.55) ITGB1ITGA4ITGB7
Hydrochloric Acid SCHEMBL5164904 0.87 ITGA4 (0.55) ITGB1ITGA4ITGB7
SCHEMBL18009483 0.83 ITGB1 (0.58) ITGB1ITGA4ITGB7GRB2SLC7A5
SCHEMBL18009482 0.83 ITGB1 (0.58) ITGB1ITGA4ITGB7GRB2SLC7A5
SCHEMBL22982364 0.80 ITGB1 (0.63) ITGB1ITGA4ITGB7GRB2PTPN1
SCHEMBL14564318 0.80 ITGA4 (0.56) ITGB1ITGA4ITGB7
SCHEMBL27504630 0.80 ITGB1 (0.62) ITGB1ITGA4ITGB7GRB2PTPN1
SCHEMBL6297453 0.80 ITGB1 (0.63) ITGB1ITGA4ITGB7GRB2PTPN1
SCHEMBL27504631 0.80 ITGB1 (0.62) ITGB1ITGA4ITGB7GRB2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1218943-C 4-pyrimidinyl-N-acyl-L-phenylalanine compounds HOFFMANN LA ROCHE (CH) 2005-09-14 CN disclosed
EP-1244625-B1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES HOFFMANN LA ROCHE (CH) 2005-06-15 EP disclosed
CN-1407972-A 4-pyrimidinyl-N-acyl-L-phenylalanine compounds HOFFMANN LA ROCHE (CH) 2003-04-02 CN disclosed
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed