SCHEMBL623881

SCHEMBL623881

FC(F)(F)c1cccc(-c2cnc3sc(NCC4CCNCC4)nn23)c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FYN P06241 9/20 0.60
MKNK1 Q9BUB5 1/20 0.56
PIM1 P11309 8/20 0.53
KDM1A O60341 1/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
KCNH2 Q12809 1/20 0.44
EPHB4 P54760 1/20 0.44
PIM3 Q86V86 1/20 0.44
PIM2 Q9P1W9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004609 0.94 FYN (0.67) FYNMKNK1PIM1KCNH2PIM3
SCHEMBL1946065 0.90 FYN (0.68) FYNMKNK1PIM1KCNH2PIM2
SCHEMBL623846 0.87 FYN (0.57) FYNMKNK1PIM1KCNH2PIM3
SCHEMBL624030 0.87 FYN (0.59) FYNMKNK1PIM1KCNH2PIM3
SCHEMBL625502 0.86 PIM1 (0.69) FYNMKNK1PIM1KCNH2PIM3
SCHEMBL625204 0.86 FYN (0.60) FYNMKNK1PIM1PIM3PIM2
SCHEMBL623851 0.83 FYN (0.61) FYNMKNK1PIM1
SCHEMBL623577 0.83 FYN (0.63) FYNMKNK1PIM1
SCHEMBL2257604 0.82 MKNK1 (0.77) FYNMKNK1PIM1
SCHEMBL628028 0.82 FYN (0.56) FYNMKNK1PIM1KCNH2PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020217-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed