SCHEMBL6240281

SCHEMBL6240281

NC(=O)CC#Cc1ccco1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.48
CYP2C19 P33261 2/20 0.39
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
NPC1 O15118 1/20 0.33
HSP90AA1 P07900 1/20 0.33
AGTR1 P30556 1/20 0.33
RAB9A P51151 1/20 0.33
PAX8 Q06710 1/20 0.33
TLR9 Q9NR96 1/20 0.33
ALDH1A1 P00352 4/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
HTT P42858 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PTPN1 P18031 1/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16345143 0.75
SCHEMBL7571198 0.75
SCHEMBL13618775 0.74 ALOX5 (0.37) ALOX5ALDH1A1
SCHEMBL11911412 0.72 ALOX5 (0.42) ALOX5CYP2C19CES2CES1NPC1
SCHEMBL6643512 0.72 ALOX5 (0.37) ALOX5CYP2C19CES2CES1ALDH1A1
SCHEMBL9906388 0.71
SCHEMBL16345466 0.71
SCHEMBL1799185 0.71 ALOX5 (0.43) ALOX5CES2CES1NPC1HSP90AA1
SCHEMBL2557403 0.69 ALOX5 (0.45) ALOX5CYP2C19CES2CES1NPC1
SCHEMBL8863670 0.69 PTPN7 (0.44) ALOX5CYP2C19ALDH1A1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077928-B1 NOVEL SUBSTITUTED CYCLIC COMPOUNDS, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2005-12-07 EP disclosed