SCHEMBL6240293

SCHEMBL6240293

CSc1ccc(C=CC(=O)O)c(Cl)c1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 8/20 0.43
ICAM1 P05362 8/20 0.43
ITGAL P20701 8/20 0.43
PTGER3 P43115 2/20 0.40
PTGER2 P43116 2/20 0.40
TBXA2R P21731 1/20 0.40
PTGDR Q13258 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
NFKB1 P19838 1/20 0.40
CA4 P22748 1/20 0.40
MIF P14174 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
ALOX5 P09917 1/20 0.37
PTGER1 P34995 1/20 0.37
PTGES O14684 1/20 0.36
HDAC3 O15379 1/20 0.36
TNKS O95271 1/20 0.36
HDAC4 P56524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6240290 1.00 ITGB2 (0.43) ITGB2ICAM1ITGALPTGER3PTGER2
SCHEMBL6817329 0.86 ITGB2 (0.52) ITGB2ICAM1ITGALPTGER3PTGER2
SCHEMBL6568833 0.86 ITGB2 (0.52) ITGB2ICAM1ITGALPTGER3PTGER2
SCHEMBL6240384 0.83 ALDH1A1 (0.44) ITGB2ICAM1ITGALCA1CA2
SCHEMBL6240387 0.83 ALDH1A1 (0.44) ITGB2ICAM1ITGALCA1CA2
SCHEMBL6310691 0.79 ITGB2 (0.39) ITGB2ICAM1ITGALPTGER3PTGER2
SCHEMBL6310686 0.79 ITGB2 (0.39) ITGB2ICAM1ITGALPTGER3PTGER2
SCHEMBL8296823 0.77 ITGB2 (0.52) ITGB2ICAM1ITGALKDM4EHTT
SCHEMBL6500029 0.77 ITGAL (0.54) ITGB2ICAM1ITGALMAPT
SCHEMBL6500024 0.77 ITGAL (0.54) ITGB2ICAM1ITGALMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019177-A1 AMINOPIPERIDINE AMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed