SCHEMBL6245293

SCHEMBL6245293

CC(C)CNC(=O)c1c[c]cc([AsH2])c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.53
KMT2A Q03164 2/20 0.53
GAA P10253 1/20 0.53
HPGD P15428 4/20 0.48
KDM4E B2RXH2 2/20 0.44
MLYCD O95822 1/20 0.44
HTT P42858 2/20 0.43
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
POLB P06746 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
TSHR P16473 1/20 0.37
MEN1 O00255 1/20 0.36
MAPK14 Q16539 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6241847 0.81 HSD17B10 (0.53) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL7579726 0.79 MLYCD (0.40) KMT2AHPGDMLYCDLMNANPSR1
SCHEMBL2908793 0.75 HSD17B10 (0.78) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL7195286 0.75 KMT2A (0.52) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL159472 0.73 KMT2A (0.63) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL7114941 0.73 HDAC6 (0.53) HSD17B10GAAHPGDLMNARAB9A
SCHEMBL17865783 0.72 MLYCD (0.73) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL27773889 0.71 KMT2A (0.61) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL6197366 0.69 CA1 (0.44) HSD17B10KMT2AGAAHPGDKDM4E
SCHEMBL1004027 0.69 GAA (0.62) HSD17B10KMT2AGAAHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268463-B1 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 4-PYRONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORP (US) 2005-02-16 EP claimed