SCHEMBL6245337

SCHEMBL6245337

Nc1cc(NC(=O)c2cc3cc(NC(=O)c4cc5c(o4)C=CC(=O)C5)ccc3[nH]2)c(CCCl)c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 6/20 0.42
PYGL P06737 7/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
NHERF1 O14745 4/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
VCP P55072 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6245333 0.82 HDAC2 (0.42) HDAC2PYGLKDM4ENPC1MAPT
SCHEMBL6242347 0.81 KDM4E (0.39) HDAC2PYGLKDM4ENPC1MAPT
SCHEMBL6248210 0.76 NPC1 (0.39) HDAC2PYGLKDM4ENPC1MAPT
SCHEMBL5733235 0.76 HDAC2 (0.47) HDAC2PYGLNHERF1TP53POLB
SCHEMBL6178778 0.74 KDM4E (0.61) KDM4ENPC1MAPTTP53
SCHEMBL6180022 0.67 KMT2A (0.43) HDAC2PYGLKDM4ENPC1MAPT
SCHEMBL5734157 0.66 TP53 (0.42) KDM4ENPC1MAPTTP53
Centanamycin SCHEMBL29441389 0.65 LMNA (0.46) KDM4EMAPTTP53POLB
Centanamycin SCHEMBL5733476 0.65 LMNA (0.46) KDM4EMAPTTP53POLB
SCHEMBL6242344 0.63 KDM4E (0.38) HDAC2PYGLKDM4ENPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320522-B1 COMPOSITIONS AND METHODS OF THE USE THEREOF ACHIRAL ANALOGUES OF CC-1065 AND THE DUOCARMYCINS TAIHO PHARMACEUTICAL CO LTD (JP) 2005-11-23 EP claimed